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Ezetimibe

Common Brand Names: Zetia

Drug Information

Medically reviewed by Jessica Swirble, PharmD
Last updated on 6/6/2024

Drug Information | Side Effects | Use & Dosage | Request a Prescription

Quick facts:
  • Brand Name: Zetia
  • Generic Name: Ezetimibe
  • Uses: Treatment for high cholesterol
  • Drug Class: Cholesterol absorption inhibitor
  • Availability: Prescription only
  • Generic Status: Yes
  • Controlled Substance: No

What is ezetimibe?

Ezetimibe is a prescription medication used to reduce high cholesterol levels in the blood. It works by blocking the absorption of cholesterol from the intestines, which helps lower LDL ("bad") cholesterol levels and raise HDL ("good") cholesterol levels.

What is ezetimibe used to treat?

Ezetimibe is typically used to treat high cholesterol and certain other lipids in the blood, such as triglycerides. It can also be used in combination with statins or other medications to treat familial hypercholesterolemia (FH), which is a genetic disorder that causes very high levels of cholesterol in the blood.

High cholesterol can lead to serious health problems, such as heart attacks and strokes. To keep cholesterol under control, ezetimibe is usually prescribed along with lifestyle changes, such as a low-cholesterol, low-saturated fat diet.

How does ezetimibe work?

Ezetimibe belongs to a class of medications known as cholesterol absorption inhibitors. These drugs work by preventing the absorption of cholesterol in the intestine. This makes it easier for your body to clear LDL cholesterol and other fats from the body.

How do I take ezetimibe?

Ezetimibe is available as an oral tablet.

The dosage and frequency of use depend on the condition being treated, its severity, and how you respond to the medication.

Follow your healthcare provider's instructions regarding dosage and schedule. Do not exceed the prescribed dose or frequency of use without consulting your provider.

How long until I see results?

Ezetimibe is used to manage high cholesterol. The effects can be noticeable within a few weeks, but it may take up to two weeks for the desired reduction in cholesterol levels to occur.

Continue using ezetimibe as prescribed, even if you start feeling better. Regular use according to your prescription is crucial for the management of your cholesterol levels.

Are there any other uses for ezetimibe?

While ezetimibe is primarily used for treating high cholesterol, healthcare providers may prescribe it off-label for other conditions.

Discuss any alternative uses of ezetimibe with your healthcare provider.

Dosage forms of ezetimibe

Ezetimibe is available in the following dosage forms:

  • Oral tablets

Ezetimibe is a prescription medication. You must have a valid prescription from a licensed healthcare provider to obtain it.