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Acyclovir

Common Brand Names: Sitavig, Zovirax

Drug Information

Medically reviewed by Jessica Swirble, PharmD
Last updated on April 17, 2025

Drug Information | Side Effects | Use & Dosage | Request an Online Prescription

Quick facts

  • Brand Name: Zovirax
  • Generic Name: Acyclovir
  • Uses: Treating viral infections such as herpes simplex, shingles, and chickenpox
  • Drug Class: Antiviral
  • Availability: Prescription only
  • Generic Status: Yes
  • Controlled Substance: No

What is acyclovir?

Acyclovir is an antiviral medication used primarily to treat infections caused by certain types of viruses. It treats cold sores around the mouth (caused by herpes simplex), shingles (caused by herpes zoster), and chickenpox.

What conditions does acyclovir treat?

Acyclovir is primarily used to treat conditions such as:

  • Herpes simplex virus infections: Helps reduce pain symptoms and speeds recovery.
  • Shingles (herpes zoster): Aids in reducing pain and the length of the infection.
  • Chickenpox: Helps reduce the length and severity of the disease.

It may also be used to treat outbreaks of genital herpes and to prevent recurrent outbreaks.

How does acyclovir work?

Acyclovir works by interfering with viral DNA synthesis, which reduces the virus's ability to replicate and spread. This helps to decrease the severity of infections and speed up the healing process.

How do I take acyclovir?

Acyclovir can be taken in different forms, depending on the specific needs:

  • Oral tablets: Typically taken several times daily.
  • Topical cream: Applied to the affected area several times a day.
  • Intravenous formulations: Used in more severe cases, administered by a healthcare provider.

The dosage and duration of treatment depend on the condition being treated, its severity, and your response to the medication.

Follow your healthcare provider's instructions regarding dosage and schedule. Do not exceed the prescribed dose or duration of treatment without consulting your provider.

How long until I feel better?

The effectiveness of acyclovir and the time it takes to notice improvement can vary among individuals. Improvement in symptoms can usually be observed within a few days of starting the medication, but it may take longer to fully recover from the infection.

Continue taking acyclovir as prescribed even if you start feeling better. Do not abruptly stop the medication, as it may lead to a return of the infection.

Are there any other uses for acyclovir?

While acyclovir is primarily used for managing viral infections, healthcare providers may sometimes prescribe it off-label for other viral infections not listed above.

Discuss any alternative uses of acyclovir with your healthcare provider.

Dosage forms of acyclovir

Acyclovir is available in the following dosage forms:

  • Oral tablets: Typically available in 400mg and 800mg dosages.
  • Oral capsules: Available in 200mg dosage.
  • Topical cream: For application to skin infections.
  • Oral suspension: Available in 200mg/5ml dosages.
  • Intravenous formulations: For severe infections.

Generic versions of acyclovir are available, providing cost-effective treatment options.

Acyclovir is a prescription medication. You will need a valid prescription from a licensed healthcare provider to obtain this medication.

Side Effects and Precautions for Acyclovir


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What are the side effects of acyclovir?

The use of acyclovir can lead to various side effects in some individuals.

Common mild side effects of acyclovir use include:

  • Headache
  • Dizziness or lightheadedness
  • Nausea or upset stomach
  • Diarrhea
  • Fatigue
  • Tiredness
  • Skin rash
  • Sensitive skin that may burn more easily in the sun
  • Vision changes

More severe side effects of acyclovir use can include:

  • Rapid heartbeat
  • Severe allergic reactions (such as rash, itching, swelling of the face, tongue, or throat, trouble breathing)
  • Changes in urine volume
  • Blood in the urine
  • Extreme tiredness
  • Easy bruising or bleeding
  • New signs of infection (like a sore throat that doesn't go away, fever)
  • Jaundice (yellowing of the skin or eyes)
  • Seizures
  • Loss of consciousness
  • Hallucinations
  • Confusion

If you experience any severe or concerning side effects while taking acyclovir, contact your healthcare provider right away.

What should I tell my healthcare provider before using acyclovir?

Tell your healthcare provider about any existing medical conditions, allergies, or other medications you are taking before starting treatment with acyclovir. This includes prescription drugs, over-the-counter medications, and dietary supplements, as they may interact with acyclovir.

Tell your provider if you are taking these medications or supplements:

  • Medications that affect kidney function
  • Antibiotics
  • Other antiviral drugs
  • Immunomodulators
  • Tizanidine
  • Nonsteroidal anti-inflammatory medications (NSAIDs)

You should also mention medical conditions such as:

  • Kidney disease
  • Liver disease
  • A weakened immune system (from HIV, bone marrow transplant, kidney transplant)
  • Neurological disorders
  • Seizure disorder
  • Hematologic disorders (problems with red blood cells, white blood cells, platelets, etc)

If you are pregnant, planning to become pregnant, or breastfeeding, consult your healthcare provider before using acyclovir to assess potential risks and benefits.

Are there any other special instructions I should follow?

Take acyclovir exactly as prescribed by your healthcare provider. Do not exceed the recommended dose or duration of treatment.

Acyclovir should be taken with or without food based on your healthcare provider's advice. It is important to follow their instructions for optimal effectiveness.

Stay hydrated while taking acyclovir, especially if you are taking higher doses, to help prevent kidney issues.

What should I do in case of an overdose?

In case of an acyclovir overdose, seek medical attention immediately. Symptoms of overdose may include agitation, loss of consciousness, and seizures. If you suspect an overdose, contact the poison control helpline at 1-800-222-1222 or call emergency services.

Proper Use & Dosage Information for Acyclovir


Drug Information | Side Effects | Use & Dosage | Request an Online Prescription

What is the typical starting dose for acyclovir?

Acyclovir is available in the following forms:

  • Oral tablets (200 mg, 400 mg, 800 mg)
  • Oral capsules
  • Suspension liquid
  • Cream
  • Ointment
  • Intravenous formulation

The typical starting dose of acyclovir varies depending on the condition being treated, the severity of symptoms, and individual patient factors. It is important to follow your healthcare provider's instructions regarding dosage and administration.

For herpes simplex virus infections, the typical starting dose may be:

  • Oral tablets: 200 mg five times daily for 10 days.

For shingles (herpes zoster), the typical dose may be:

  • Oral tablets: 800 mg five times daily for 7 to 10 days.

The dosage may be adjusted based on the response and tolerance to the medication. Your healthcare provider will determine the most appropriate dose based on your medical history, current medications, and response to the medication.

Acyclovir should be taken exactly as prescribed by your healthcare provider. Do not exceed the recommended dose or duration of treatment without consulting your provider.

If you have any questions about your dosage or need adjustments, contact your healthcare provider for guidance. If you need immediate medical advice or assistance, consider scheduling an online doctor appointment through a platform like Sesame.

What should I do if I miss a dose of acyclovir?

If you miss a dose of acyclovir, take it as soon as you remember unless it is close to the time for your next scheduled dose. In that case, skip the missed dose and continue with your regular dosing schedule. Do not double the dose to make up for a missed one.

Maintain a consistent dosing schedule to ensure the effectiveness of acyclovir in managing your viral infection.

What should I do if I'm feeling better while taking acyclovir?

Continue taking acyclovir as prescribed by your healthcare provider, even if you start feeling better. Do not stop the medication abruptly without consulting your provider, as it may lead to a recurrence of symptoms or other complications.

Complete the full course of treatment as directed to minimize the risk of relapse.

If you have any concerns or questions about your medication, discuss them with your healthcare provider for personalized guidance and recommendations.

How should I store acyclovir?

Store acyclovir according to the instructions provided by your healthcare provider or pharmacist. Keep it at room temperature, away from moisture, heat, and light. Ensure the container is tightly closed and out of reach of children.

Do not use expired medication or medications that appear damaged or discolored. If you have any questions about storage, consult your healthcare provider or pharmacist for guidance.

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