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Bupropion

Common Brand Names: Aplenzin, Forfivo, Wellbutrin, Zyban

Drug Information

Medically reviewed by Jessica Swirble, PharmD
Last updated on April 2, 2025

Drug Information | Side Effects | Use & Dosage | Request an Online Prescription

Quick facts

  • Brand Name: Aplenzin, Forfivo, Wellbutrin, Zyban
  • Generic Name: Bupropion
  • Uses: Depression, SAD, smoking cessation
  • Drug Class: Norepinephrine-dopamine reuptake inhibitor (NDRI)
  • Availability: Prescription only
  • Generic Status: Yes
  • Controlled Substance: No

What is bupropion?

Bupropion is an antidepressant medication that belongs to the class of drugs known as norepinephrine-dopamine reuptake inhibitors (NDRIs). It is used to treat major depressive disorder (MDD), and seasonal affective disorder (SAD). It is also used to help in smoking cessation (quitting smoking).

What conditions does bupropion treat?

Bupropion is used to treat conditions such as:

  • Major depressive disorder (MDD)
  • Seasonal affective disorder (SAD)
  • Smoking cessation (as part of a comprehensive smoking cessation program)

It may also be prescribed for other mental health conditions or off-label uses as determined by your healthcare provider.

How does bupropion work?

Bupropion works by increasing levels of norepinephrine and dopamine, two neurotransmitters in the brain that are involved in regulating mood and behavior.

How do I take bupropion?

Bupropion is usually taken orally with or without food, as directed by your healthcare provider.

Regular bupropion is taken three times a day (every 6 hours) or four times a day (every 4 hours). Sustained-release bupropion is taken twice a day, and extended-release bupropion is taken once a day (usually in the morning).

The dosage and duration of bupropion treatment depend on your condition and response to the medication. Patients taking bupropion for seasonal affective disorder are usually ordered to start taking it in the fall, continue it through the winter, and stop taking it in the spring.

Follow the prescribed dosage and schedule strictly. Do not stop taking bupropion suddenly without consulting your healthcare provider, as it may cause withdrawal symptoms.

How long until I feel better?

The time it takes to feel the full effects of bupropion can vary from person to person. Some people may notice improvement in their symptoms within a few weeks, while others may require several weeks of treatment.

It's important to continue taking bupropion as prescribed even if you do not feel better immediately. Talk to your healthcare provider if you have any concerns about your treatment.

Are there other uses for bupropion?

While bupropion is primarily used for depression, SAD, and smoking cessation, healthcare providers may sometimes prescribe it off-label for other conditions, such as:

  • Attention deficit hyperactivity disorder (ADHD)
  • Depression in patients with bipolar disorder

Discuss any alternative uses of bupropion with your healthcare provider.

Dosage forms of bupropion

Bupropion is available in the following dosage forms:

  • Oral tablets: Available in various strengths (e.g., 75mg, 150mg, 300mg)
  • Extended-release oral tablets
  • Oral sustained-release tablets

Generic versions of bupropion are available under various brand names.

Bupropion is a prescription medication. You will need a valid prescription from a licensed healthcare provider to obtain this antidepressant.

Side Effects and Precautions for Bupropion


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What are the side effects of bupropion?

The use of bupropion can lead to various side effects in some individuals.

Common mild side effects of bupropion use include:

  • Nausea
  • Dry mouth
  • Sore throat
  • Headache
  • Constipation
  • Insomnia or drowsiness
  • Increased sweating
  • Increased urination
  • Anxiety or excitement
  • Tremors (uncontrollable shaking)
  • Changes in appetite or weight
  • Dizziness
  • Blurred vision
  • Ringing in the ears
  • Changes in taste
  • Increased heart rate

More severe side effects of bupropion use can include:

  • Seizures (especially at higher doses)
  • Suicidal thoughts or behavior (especially in young adults)
  • Agitation or restlessness
  • Manic episodes (abnormally high energy, racing thoughts, reckless behavior)
  • Hallucinations
  • Irregular heartbeat
  • Severe allergic reactions (rash, itching/swelling, severe dizziness, trouble breathing)

If you experience any severe side effects while taking bupropion, seek immediate medical attention.

What should I tell my healthcare provider before using bupropion?

Inform your healthcare provider about any existing medical conditions, allergies, or other medications you are taking before starting treatment with bupropion. This includes prescription drugs, over-the-counter medications, and dietary supplements, as they may interact with bupropion.

Tell your provider if you are taking these medications or supplements:

  • MAO inhibitors (e.g., selegiline, phenelzine)
  • Other antidepressants (e.g., SSRIs, SNRIs, tricyclic antidepressants)
  • Antipsychotics
  • Anti-seizure medications
  • Blood thinners (e.g., warfarin)
  • Stimulants
  • Herbal supplements (e.g., St. John's wort)

Mention medical conditions such as:

  • History of seizures or epilepsy
  • Bipolar disorder or mania
  • Eating disorders
  • Liver or kidney disease
  • High blood pressure
  • Heart disease
  • Diabetes
  • Glaucoma
  • Alcohol or substance use disorder

If you are pregnant, planning to become pregnant, or breastfeeding, consult your healthcare provider before using bupropion to assess potential risks and benefits.

Are there any other special instructions I should follow?

Take bupropion exactly as prescribed by your healthcare provider. Do not increase or decrease the dosage without consulting them.

It may take several weeks for bupropion to take full effect. Continue taking the medication even if you do not immediately feel better.

Avoid alcohol while taking bupropion, as it may worsen certain side effects and increase the risk of seizures.

Do not suddenly stop taking bupropion without your healthcare provider's guidance, as it may cause withdrawal symptoms.

What should I do in case of an overdose?

In case of a bupropion overdose, seek immediate medical attention. Symptoms may include seizures, hallucinations, rapid heart rate, fainting, and loss of consciousness. If you suspect an overdose, contact the poison control helpline at 1-800-222-1222 or call emergency services.

Proper Use & Dosage Information for Bupropion


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What is the typical starting dose for bupropion?

Bupropion is available in various strengths, including:

  • Oral tablets (75 mg, 100 mg)
  • Extended-release tablets (150 mg, 300 mg, 450 mg)
  • Sustained-release tablets (100 mg, 150 mg, 200 mg)

The typical starting dose of bupropion for depression, seasonal affective disorder (SAD), smoking cessation, and other conditions can vary depending on factors such as the specific condition being treated, your age, other medical conditions, and how you respond to the medication. It's crucial to follow your healthcare provider's instructions regarding dosage and administration carefully.

For most adults with depression or SAD, the typical starting dose of bupropion may be:

  • 100 mg taken orally twice daily for immediate-release tablets
  • 150 mg taken orally once daily for extended-release tablets and sustained-release tablets

For smoking cessation, the typical starting dose of bupropion may also be:

  • 150 mg taken orally once daily for sustained-release tablets

However, your healthcare provider may start with a lower dose, such as 75 mg for immediate-release tablets, especially for older adults or those with certain medical conditions. The dose may then be gradually increased based on your response and tolerability, up to a maximum of 400 mg (for sustained-release) to 450 mg (for extended-release) per day for depression and 300 mg per day for SAD and smoking cessation.

Bupropion can be taken with or without food, but it's important to take it consistently at the same time each day.

Your healthcare provider will monitor your response to bupropion and may adjust the dose as needed. It's important not to exceed the recommended dose or make changes to your dosage without consulting your healthcare provider.

If you have any questions about your dosage or how to take bupropion, contact your healthcare provider or pharmacist. If you want to talk to a provider right away, consider booking an online doctor appointment on Sesame to discuss your concerns.

What should I do if I miss a dose of bupropion?

If you miss a dose of bupropion, take it as soon as you remember. If it's close to the time for your next dose, skip the missed dose and continue with your regular dosing schedule. Avoid taking a double dose of bupropion to make up for a missed one.

What should I do if I'm feeling better while taking bupropion?

Continue taking bupropion as prescribed by your healthcare provider, even if you start feeling better. Abruptly stopping bupropion can lead to withdrawal symptoms and potential relapse of symptoms. Follow your provider's instructions regarding the duration of treatment.

How should I store bupropion?

Store bupropion according to the instructions provided by your healthcare provider or pharmacist. It should be kept at room temperature, away from excessive heat, light, and moisture. Ensure the container is tightly closed and keep the medication out of the reach of children.

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